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Toceranib phosphate

Toceranib phosphate

商品货号:CC5428 用户评价: comment rank 5

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¥517.00元
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产品描述:

Toceranib phosphate, the phosphate salt of toceranib, is a selective inhibitor of the tyrosine kinase activity of several members of the split kinase RTK family, including Flk-1/KDR, PDGFR, and Kit with Ki values of 6 nM and 5 nM for Flk-1/KDR and PDGFRβ, respectively.

化学数据:

分子量Molecular Weight (MW) 494.45
化学式Formula

 

C22H25FN4O2.H3O4P

 

CAS号CAS No. 874819-74-6
溶解性Solubility (25°C) *  二甲基亚砜DMSO 2 mg/mL(4.04 mM)
水Water 2 mg/mL(4.04 mM)
乙醇Alcohol Insoluble


制备储备液

浓度 溶剂体积(DMSO) 质量 1 mg 5 mg 10 mg
1 mM 2.0224 mL 10.1122 mL 20.2245 mL
5 mM - - -
10 mM - - -
50 mM - - -


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